References

1. Hill, S.J., Baker, J.G., Rees, S. (2001) Reporter-gene systems for the study of G-protein- coupled receptors. Curr Opin Pharmacol. 1, 526-532.

2. Windh, R.T., Manning, D.R. (2002) Analysis of G protein activation in Sf9 and mammalian cells by agonist-promoted [35S]GTPyS binding. Methods Enzymol. 344, 3-14.

3. Milligan, G. (2003) Principles: Extending the utility of [35S]GTPyS binding assays. Trends Pharmacol Sci. 24, 87-90.

4. Harrison, C., Traynor, J.R. (2003) The [35S]GTPyS binding assay: Approaches and applications in pharmacology. Life Sci. 74 , 489 - 508 .

5. Fang, Y., Lahiri, J., Picard, L. (2003) G protein-coupled receptor microarrays for drug discovery. Drug Discov Today. 8 , 755 - 761 .

6. Waller, A. , Simons, P.C. , Biggs, S.M. , Edwards, B.S. , Prossnitz , E.R. , Sklar, L.A. (2004) Techniques: GPCR assembly, pharmacology and screening by flow cytometry. Trends Pharmacol Sci. 25, 663-669.

7. Kenakin, T. (ed) (1993) Pharmacological Analysis of Drug-Receptor Interactions. New York: Raven.

8. Limberd, L.E. (1996) Cell surface receptors: A Short Course on Theory and Methods, 2nd ed. Boston: Martinus Nijhoff.

9. Bylund, D.B.,Toews, M.L. (1993) Radioligand binding methods: Practical guide and tips. Am J Physiol. 265 , L421 - L429 .

10. Muramatsu, I., Tanaka, T., Suzuki, F., Li, Z., Hiraizumi-Hiraoka, Y., Anisuzzaman, A.S., Yamamoto, H., Horinouchi, T., Morishima, S. (2005) Quantifying receptor properties: The tissue segment binding method—A powerful tool for the pharma-come analysis of native receptors. J Pharmacol Sci. 98, 331-339.

11. Mazzoni, M.R., Martini, C., Lucacchini, A. (1993) Regulation of agonist binding to A2A adenosine receptors: Effects of guanine nucleotides (GDPPS and GTPyS) and Mg2+ ion. Biochim Biophys Acta. 1220, 76-84.

12. Rosenthal, H.E. (1967) A graphic method for the determination and presentation of binding parameters in a complex system. Anal Biochem. 20 , 525 - 532 .

13. Cheng, Y., Prusoff, W.H. (1973) Relationship between the inhibition constant (K;) and the concentration of inhibitor which causes 50 per cent inhibition (IC50) of an enzymatic reaction . Biochem Pharmacol. 22, 3099-3108.

14. Motulsky, H.J. (1999) The complete guide to nonlinear regression. Published online by GraphPad Software. http://www.curvefit.com.

15. Bylund, D.B. (1986) Graphic presentation and analysis of inhibition data from ligand-binding experiments. Anal Biochem. 159, 50-57.

16. Carpenter, J.W., Laethem, C., Hubbard, F.R., Eckols, T.K., Baez, M., McClure, D., Nelson, D.L., Johnston, P.A. (2002) Configuring radioligand receptor binding assays for HTS using scintillation proximity assay technology. Methods Mol Biol. 190 , 31 - 49 .

17. Sutherland, E.W., Rall, T.W. (1958) Fractionation and characterization of a cyclic adenine ribonucleotide formed by tissue particles. J Biol Chem. 232,1077-1091.

18. Williams, C. (2004) cAMP detection methods in HTS: Selecting the best from the rest. Nat Rev Drug Discov. 3,125-135.

19. Salomon, Y. (1979) Adenylate cyclase assay. Adv Cyclic Nucleotide Res. 10, 35-55.

20. Salomon, Y., Londos, C., Rodbell, M. (1974) A highly sensitive adenylate cyclase assay. Anal Biochem. 58, 541-548.

21. Johnson, R.A., Salomon, Y. (1991) Assay of adenylyl cyclase enzymatic activity. Methods Enzymol. 195 , 3 - 21 .

22. Post, S.R., Ostrom, R.S., Insel, P.A. (2000) Biochemical methods for detection and measurement of cyclic cAMP and adenylyl cyclase activity. Methods Mol Biol. 126 , 363 - 374 .

23. Wiegn, P., Dutton, J., Lurie, K.G. (1993) An enzymatic fluorimetric assay for adenylate cyclase activity. Anal Biochem. 208, 217-222.

24. Sugiyama, A., Lurie, K.G. (1994) An enzymatic fluorimetric assay for adenosine 3':5'-monophosphate. Anal Biochem. 218, 20-25.

25. Sugiyama, A., McKnite, S., Lurie, K.G. (1995) Measurement of adenylylcyclase activity with an enzymatic fluorimetric assay. Anal Biochem. 225, 368-371.

26. Lowry, O.H., Passonneau, J.V. (1972) A Flexible System ofEnzymatic Analysis. New York : Accademic.

27. McKnite, S., Evingson, M., Pennington, J., Adkisson, W., Sugiyama, A., Lurie, K.G. (1996) A bioluminescent enzymatic assay for adenylylcyclase activity. Anal Biochem. 235 , 103 - 106 .

28. Kumar, M., Hsiao, K., Vidugiriene, J., Goueli, S.A. (2007) A bioluminescent-based, HTS-compatible assay to monitor G-protein-coupled receptor modulation of cellular cAMP. Assay Drug Dev Technol. 5 , 237 - 245 .

29. Steiner, A.L., Kipnis, D.M., Utiger, R., Parker, C. (1969) Radioimmunoassay for the measurement of adenosine 3',5'-cyclic monophosphate. Proc Natl Acad Sci USA. 64, 367-373.

30. Harper, J.F., Brooker, G. (1975) Femtomole sensitive radioimmunoassay for cyclic AMP and cyclic GMP after 2'0 acetylation by acetic anhydride in aqueous solution. J Cyclic Nucleotide Res. 1, 207-218.

31. Brooker, G., Harper, J.F.,Terasaki, W.L., Moylan, R.D. (1979) Radioimmunoassay of cyclic AMP and cyclic GMP. Adv Cyclic Nucleotide Res. 10 , 1 - 33 .

32. Daniels, C.K., Zhang, L., Musser, B., Vestal, R.E. (1994) A solid-phase radioimmunoassay for cyclic AMP. J Pharmacol Toxicol Methods. 31,41-46.

33. Yamamoto, I., Tsuji, J. (1981) Enzyme immunoassay of cyclic adenosine 5', 5'-monophosphate (AMP) using ß-D-galactosidase as label. Immunopharmacology. 3 , 53 - 59 .

34. Pradelles, P., Grassi, J., Chabardes, D., Guiso, N. (1989) Enzyme immunoassays of adenosine cyclic 3',5'-monophosphate and guanosine cyclic 3',5'-monophosphate using acetylcholinesterase. Anal Chem. 61,447-453.

35. Linden, J., Vandenhoff, G.E., Taylor, D., Finkelstein, G.L. (1992) Solid phase enzyme immunoassay of cyclic adenosine 3',5'-monophosphate. Effect of coating strategy upon assay performance in comparison with radioimmunoassay. J Immunol Methods. 151 , 209 - 216 .

36. Tsugawa, M., Iida, S., Fujii, H., Moriwaki, K., Tarui, S., Sugi, M., Yamane, R., Fujimoto, M. (1990) An enzyme-linked immunosorbent assay (ELISA) for adenosine 3',5'-cyclic monophosphate (cAMP) in human plasma and urine using monoclonal antibody. J Immunoassay. 11,49-61.

37. Gilman, A.G. (1970) A protein binding assay for adenosine 3':5'-cyclic monophosphate. Proc Natl Acad Sci U S A. 67, 305-312.

38. Brown, B.L., Albano, J.D.M., Ekins, R.P., Sgherzi, A.M. (1971) A simple and sensitive saturation assay method for the measurement of adenosine 3' :5'-cyclic monophosphate. Biochem J. 121, 561-562.

39. Santa Coloma,T.A., Bley, M.A., Charreau, E.H. (1987) Improvement on the competitive binding assay for the measurement of cyclic cAMP by using ammonium sulphate precipitation . Biochem J. 245, 923-924.

40. Takeda, T., Kuno, T., Shuntoh, H., Tanaka, C. (1989) A rapid filtration assay for cAMP. J Biochem. 105, 327-329.

41. Nordstedt, C., Fredholm, B.B. (1990) A modification of protein binding method for rapid quantification of cAMP in cell-culture supernatants and body fluid. Anal Biochem. 189, 231-234.

42. Kuo, J.F., Greengard, P. (1970) Cyclic nucleotide-dependent protein kinases. An assay method for the measurement of adenosine 3',5'-monophosphate in various tissues and a study of agents influencing its level in adipose cells. J Biol Chem. 245, 4067 - 4073 .

43. Wastila , W.B. , Stull , J.T. , Mayer, S.E. , Walsh , D.A. ( 1971 ) Measurement of cyclic 3' ,5'-adenosine monophosphate by the activation of skeletal muscle protein kinase. J Biol Chem. 246,1996-2003.

0 0

Post a comment