References

[ 1] Haggerty, W. J., and Murrill, E. A., Res. Dev. 25, 30 (1974)

[ 2] Henry, D., Block, J. H., Anderson, J. L., and Carlson, G. R., J. Med. Chem.19, 619-626 (1976)

[ 3] Mirrlees, M. S., Moulton, S. J., Murphy, C. T., and Taylor, P. J., J. Med. Chem. 19, 615-619 (1976)

[ 4] Unger, S. H., Cook, J. R., and Hollenberg, J. S, J. Pharm. Sei. 67, 1364-1366 (1978)

[ 5] Kaliszan, R., J. Chromatogr. 220, 71-83 (1981)

[ 6] Lambert, W. J., 7. Chromatogr. A 656, 469-484 (1993)

[ 7] Braumann, Th., Weber, G., and Grimme, L. H., J. Chromatogr. 261, 329-343 (1983)

[ 8] El Tayar, N., Van de Waterbeemd, H., and Testa, B., 7. Chromatogr. 320, 293-304 (1985)

[ 9] ElTayar, N., Van de Waterbeemd, H., and Testa, B., J. Chromatogr. 320, 305-312 (1985)

[10] Reymond, D., Chung, G. N., Mayer, J. M., and Testa, B., J. Chromatogr. 391, 97-109 (1987)

[11] Valko, K., Snyder, L. R., and Glajch, J. L., J. Chromatogr. A 656, 501-520 (1993)

[12] Schoenmakers, P. J., Billiet, H. A. H., and De Galan, L., J. Chromatogr. 185, 179-195 (1979)

[13] Hsieh, M.-M., and Dorsey, J. G., J. Chromatogr. 631, 63-78 (1993)

[14] Horvath, C., Melander, W., and Molnar, I., J. Chromatogr. 125, 129-156 (1976)

[15] Wells, M. J. M., and Clark, R., J. Chromatogr. 284, 319-355 (1984)

[16] Valko, K., and Siegel, P., J. Chromatogr. 631, 49-61 (1993)

[17] ElTayar, N., Van de Waterbeemd, H., and Testa, B., Quant. Struct.-Act. Relat. 4, 69-77 (1985)

[18] Yamagami, C., Yokota, M., andTakao, N., J. Chroamtogr. A 662, 49-60 (1994)

[19] Yamagami, C., Yokota, M. andTakao, N., Chem. Pharm. Bull. 42, 907-912 (1994)

[20] Tan, L. C., and Carr, P. W., J. Chromatogr. A 656, 521-535 (1993)

[21] Kalizan, R., Quant. Struct.-Act. Relat. 9, 83-87 (1990)

[22] Rippel, G., Alattyani, E., and Szepesy, L., J. Chromatogr. A 668, 301-312 (1994)

[23] Miyake, K., andTerade, H., J. Chromatogr. 157, 386-390 (1978)

[24] Taylor, P. J. Hydrophobic properties of drugs. In: Comprehensive Medicinal Chemistry, Vol. 4. Hansch, C., Sammes, P. G. and Taylor, J. B. (Eds.). Pergamon Press: Oxford; 241-294 (1990)

[25] El Tayar, N., Tsantili-Kakoulidou, Röthlisberger, T., Testa, B., and Gal, J., J. Chromatogr. 439, 237-244 (1988)

[26] Pagliara, A., Khamis, E., Trinh, A., Carrupt, P.-A.,Tsai, R.-S. andTesta, B.,]. Liq. Chromatogr. 18, 1721-1745 (1995)

[27] Kansy, M., Fischer, H. and Van de Waterbeemd, H., Correlations between log P and RP-HPLC log k„ values: effect of charge and conformation. In: Trends in QSAR and Molecular Modeling 94. Sanz, F. (Ed.). Prouse: Barcelona 1995

[28] Van de Waterbeemd, H., Karajiannis, H., Kansy, M., Obrecht, D., Müller, K., and Lehmann, Chr., Conformation-lipophilicity relationships of peptides and peptide mimetics. In: Trends in QSAR and Molecular Modeling 94. Sanz, F. (Ed.). Prouse: Barcelona 1995

[29] Altomare, C., Cellamera, S., Carotti, A., and Ferappi, M., Quant. Struct.-Act. Relat. 12, 261-268 (1993)

[30] Miyake, K., andTerada, H., J. Chromatogr. 240, 9-20 (1982)

[31] Vallat, P., Fan, W., El Tayar, N., Carrupt, P.-A., and Testa, B., J. Liq. Chromatogr. 15, 2133-2151 (1992)

[32] Altomare, C.,Tsai, R.-S., ElTayar, N.,Testa, B., Carotti, A., Cellamare, S., and De Bene-detti, P. G., J. Pharm. Pharmacol. 43, 191-197 (1991)

[33] Miyake, K., Kitaura, F., Mizuno, N., and Terada, H., Chem. Pharm. Bull. 35, 377-388 (1987)

[34] Rothemund, S., Krause, E., Ehrlich, A., Bienert, M., Glusa, E. and Verhallen, P., J. Chromatogr. A. 661, 77-82 (1994)

[35] Haky, J. E. and Vemulapalli, S., J. Liq. Chromatogr. 13, 3111-3131 (1990)

[36] Miyake, K., Kitaura, F., Mizuno, N. andTerada, H., J. Chromatogr. 389, 47-56 (1987)

[37] Ong, S., Cai, S.-J., Bemal, C., Rhee, D., Qui, X., and Pidgeon, C., Anal. Chem. 66, 782-792 (1994)

[38] Kaliszan, R., Nasal, A., and Bucinski, A., Eur. J. Med. Chem. 29, 163-170 (1994)

[39] Pidgeon, C., Ong, S., Liu, H., Qui, X., Pidgeon, M., Dantzig, A. H., Munroe, J., Hornback, W. J., Kasher, J. S., Glunz, L., and Szczerba, T., J. Med. Chem. 38, 590-594 (1995)

[40] Ong, S., Liu, H., Qiu, X., Bhat, G., and Pidgeon, C.,Anal. Chem. 67, 755-762 (1995)

[41] Kaibara, A., Hohda, C., Hirata, N., Hirose, M., and Nakagawa, T., Chromatographia 29, 275-288 (1990)

[42] Tanaka, A., Nakamura, K., Nakanishi, I., and Fujiwara, H., J. Med. Chem. 37, 4563-4566 (1994)

[43] Van de Waterbeemd, H., and Testa, B., Adv. Drug Res. 16, 85-225 (1987)

[44] Horvath, C., Melander, W. and Molnar, I., J. Anal. Chem. 49, 142-154 (1977)

[46] Belsner, K., Pfeifer, M., and Wilfert, B., J. Chromatogr. 629, 123-134 (1993)

[47] Rodgers, A. H., and Khaledi, M. G.,Anal. Chem. 66, 327-334 (1994)

[48] Zou, H., Zhang, Y., Hong, M., and Lu, P., J. Chromatogr. 625, 169-175 (1992)

[49] Martorell, C., Calpena, A. C., Escribano, E., and Pöblet, J. M., J. Chromatogr. A. 655, 177-184 (1993)

[50] Carr, P. W., Martire, D. E., and Snyder, L. R., Special issue on the retention process in reversed-phase liquid chromatography, /. Chromatogr. 656A, 1-616 (1993)

[51] Hanai, T., J. Liq. Chromatogr. 16, 1453-1462 (1993)

[53] Cheong, W. J., and Carr, P. W„Anal. Chem. 61, 1524-1529 (1989)

[54] Rosés, M., and Bosch, E., Anal. Chim. Acta 274, 147-162

[55] Hellai, F., Phan-Tan-Luu, R., and Siouffi, A. M., J. Liq. Chromatogr. 17, 2845-2869 (1994)

[56] Park, J. H., Chae, J. J., Nah, T. H., and Jang, M. D.,J. Chromatogr. A 664, 149-158 (1994)

[57] Helburn, R. S., Rufan, S. C., Pompano, J., Mitchem, D., and Patterson, W. T., Anal. Chem. 66, 610-618 (1994)

[58] Tan, L. C., Carr, P. W., Fréchet, J. M. J., and Smigol, V., Anal. Chem. 66, 450-457 (1994)

[59] Minick, D. J., Brent, D. A., and Frenz, J., J. Chromatogr. 461, 177-191 (1989)

[60] Chen, N., Zhang, Y., and Lu, P., J. Chromatogr. 633, 31-41 (1993)

[61] El Tayar, N., Karajiannis, H., and Van de Waterbeemd, H., Amino Acids 8,125-139 (1995)

[62] Büttner, K., Ostresh, J. M., and Houghten, R. A., Induced conformational effects during RPHPLC: Prediction of immunodominant TH-cell antigenic sites. In: Peptides. Chemistry, Structure and Biology. Rivier, J. E., and Marshall, G. R. (Eds.). Escom: Leiden; 423-425 (1990)

[63] Lee, D. W., and Cho, B. Y., J. Liq. Chromatogr. 17, 2541-2558 (1994)

[64] Harnisch, M., Möckel, H. J., and Schulze, G., J. Chromatogr. 282, 315-332 (1983)

Lipophilicity in Drug Action and Toxicology edited by Vladimir PliSka,Bernard Testa & Han van de Waterbeemd Copyright© VCH Verlagsgesellschaft mbH,1996

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